| Isolate | Bark source | Researched activity | 
| Paclitaxel, taxanes | Taxus | chemotherapeutic | 
| Paeonol | Paeonia suffruticosa | various | 
| Honokiol, 4-O-methylhonokiol, magnolol, obovatol | Magnolia | neurotrophic & anti-inflammatory | 
| Salicylic acid | Salix alba | antipyretic, analgesic | 
| Yohimbine, corynanthine, ajmalicine, rauwolscine | west African evergreen | MAOI, stimulant | 
| beta-carbolines, harmala alkaloids | numerous | MAOI | 
| Cinnamon, camphor, cinnamaldehyde | Cinnamomum | blood sugar stabilizer, antioxidant | 
| Quinine, quinidine, cinchonidine, cinchonine | Cinchona | antipyretic, analgesic, antimalarial | 
| Safrole | Sassafras |  | 
| Huáng bǎi | Amur cork tree (Phellodendron amurense) | TCM | 
| Strictamine | Alstonia scholaris |  | 
|  | Slippery Elm (Ulmus rubra) | demulcent | 
| Geniposidic acid | Eucommia ulmoides |  | 
| N-methyltryptamine, serotonin analogs | numerous species from Brazil, Mexico, Taiwan | serotonin agonist, neuroimmunologic modulator | 
| Quassin | Quassia amara | various | 
| Celastrol | Tripterygium wilfordii | various | 
| Mitraphylline | Cat's claw (Uncaria tomentosa) | anti-inflammatory | 
| Ellagic acid, rutin, gallic acid, ethyl gallate | Ailanthus altissima | various | 
| Coronaridine, voacangine, ibogamine, ibogaine, tabernanthine | Voacanga africana, Tabernanthe iboga | neuroimmunologic modulator | 
| Lapachol, quercetin | Pau D'Arco (Handroanthus impetiginosus) | therapeutic naphthoquinone | 
| Icariin | Eucommia | PDE5 inhibitor | 
| Baicalin | Oroxylum indicum | prolyl endopeptidase inhibitor | 
| Frankincense, incensole | Boswellia sacra, Boswellia | incensole is a TRPV3 agonist | 
| QS21 | Quillaja saponaria (soap bark tree) | potential immunologic adjuvant | 
| Sandalwood oil, α-Santalol, β-Santalol | Sandalwood (Santalum) | Ayurvedic component | 
| Bergenin, α-viniferin, ε-viniferin, diptoindonesin A | Bergenia ligulata, Dryobalanops aromatica, Mallotus japonicus | component of Ayurvedic medicine "Paashaanbhed" | 
| Phenolic lactones | Caesalpinia paraguariensis | component of Bolivian traditional medicine | 
| Erythravine | Erythrina mulungu | Brazilian medicinal plant | 
| Antimicrobial, anti-inflammatory compounds | Psidium guajava (Guava tree) | component of traditional medicine | 
| Perfume resin | Agarwood / Oud Wood | aromatherapy | 
| Opopanax, balsam, bdellium, bisabol | Myrrh (Commiphora) | component of Eastern-Mediterranean, Middle-Eastern, and North-African, traditional medicine | 
| Rotenoids, piscidone | Jamaican dogwood (Piscidia piscipula) | component of Caribbean traditional medicine | 
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